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Product Name: Linsitinib
Chemical Name: (1r,3r)-3-(8-amino-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl)-1-methylcyclobutanol
SMILES Code: O[C@@]1(C)C[C@H](C2=NC(C3=CC=C4C=CC(C5=CC=CC=C5)=NC4=C3)=C6C(N)=NC=CN62)C1
CAS NO: 34041-84-4 Product: PFI-3
Synonym: OSI 906; OSI-906; OSI906
Chemical Formula: C26H23N5OMolecular Weight: 421.49
Appearance: Solid powderMedchemexpress.com
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Vitamin D Related inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: Linsitinib (OSI-906) is highly potent, orally efficacious and highly selective, dual ATP-competitive inhibitor of IGF-1R (IC50= 35 nM) and insulin receptor (IC50=75 nM).PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/7966611

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Author: DNA_ Alkylatingdna