Product Name :
BIM 23056
CAS NO. :
150155-61-6
Formula :
C83H96N13O17
Molecular Weight::
1547.73
Target:
Somatostatin Receptor
Serial Number:
Asp-Phe-Phe-Tyr-Asp-Trp-Lys-Val-Phe-Asp-2Nal-NH2
Short serial number :
DFFYDWKVFD-2Nal-NH2
Purity:
95%
Description :
BIM 23056 acetate is a potent and surmountable human recombinant somatostatin receptor antagonist (Ki = 142, >1000, 10.8, 16.6 and 5.7 nM for human cloned sst1-5 receptors, respectively). It acts as an antagonist on SRIF14-induced [35S]-GTPγS binding at sst3 and sst5 receptors (PKB = 6.33 and 5.84, respectively).
References:
[1]. Y C Patel, et al. Subtype selectivity of peptide analogs for all five cloned human somatostatin receptors (hsstr 1-5). Endocrinology. 1994 Dec;135(6):2814-7. [2]. W Feniuk, et al. Further evidence from functional studies for somatostatin receptor heterogeneity in guinea-pig isolated ileum, vas deferens and right atrium. Br J Pharmacol. 1995 Jul;115(6):975-80.
Related websites: https://www.medchemexpress.com/antibodies.html
Popular product recommendations:
TBK1 Antibody (YA040)
Phospho-mTOR (Ser2448) Antibody (YA171)
Cleaved-Caspase 3 p12 Antibody: Cleaved-Caspase 3 p12 Antibody is a non-conjugated and Rabbit origined monoclonal antibody about 32 kDa, targeting to Cleaved-Caspase 3 p12. It can be used for WB,ICC/IF assays with tag free, in the background of Human, Mouse, Rat.
