Product Name: SCH772984
Chemical Name: (R)-1-(2-oxo-2-(4-(4-(pyrimidin-2-yl)phenyl)piperazin-1-yl)ethyl)-N-(3-(pyridin-4-yl)-1H-indazol-5-yl)pyrrolidine-3-carboxamide
SMILES Code: O=C([C@H]1CN(CC(N2CCN(C3=CC=C(C4=NC=CC=N4)C=C3)CC2)=O)CC1)NC5=CC6=C(NN=C6C7=CC=NC=C7)C=C5
CAS NO: 179474-85-2 Product: Gilteritinib
Synonym: SCH 772984; SCH-772984
Chemical Formula: C33H33N9O2
Appearance: Solid powderWeb Site click
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).PKD inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: SCH772984 potently inhibits ERK1 and ERK2 activity with IC50 values of 4 and 1 nM, respectively. SCH722984 showed activity against BRAF mutant, NRAS mutant and wild-type melanoma.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/12414725
