Product Name: Palosuran
Chemical Name: 1-[2-(4-benzyl-4-hydroxypiperidin-1-yl)ethyl]-3-(2-methylquinolin-4-yl)urea
SMILES Code: CC1=NC2=CC=CC=C2C(=C1)NC(=O)NCCN3CCC(CC3)(CC4=CC=CC=C4)O
CAS NO: 1403783-31-2 Product: Pirarubicin (Hydrochloride)
Synonym: ACT058362; ACT 058362; ACT-058362
Chemical Formula: C25H30N4O2
Appearance: Solid powderWeb Site click
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Vasopressin Receptor inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: Palosuran (ACT058362) is a nonpeptidic, potent and selective antagonist of the urotensin-II receptor. It is selective toward human receptor. The IC50 value of it to rat receptor is 1475nM. The efficacy of palosuran to inhibit Ca2+ mobilization in CHO cellPubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/16150925