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Product Name: PIK-294
Chemical Name: 2-((4-amino-3-(3-hydroxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one
SMILES Code: O=C1N(C2=CC=CC=C2C)C(CN3N=C(C4=CC=CC(O)=C4)C5=C(N)N=CN=C53)=NC6=C1C(C)=CC=C6
CAS NO: 205304-86-5 Product: Sivelestat (sodium)
Synonym: PIK294; PIK 294
Chemical Formula: C28H23N7O2Molecular Weight: 489.52792
Appearance: Solid powderMedchemexpress.com
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).Drug-Linker Conjugates for ADC inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: PIK-294 is a highly selective p110δ inhibitor with IC50 of 10 nM, 1000-, 49- and 16-fold less potent to PI3Kα/β/γ, respectively.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/18559613

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Author: DNA_ Alkylatingdna