Product Name: GSK 525762A
Chemical Name: 2-[(4S)-6-(4-chlorophenyl)-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide
SMILES Code: CCNC(=O)CC1C2=NN=C(N2C3=C(C=C(C=C3)OC)C(=N1)C4=CC=C(C=C4)Cl)C
CAS NO: 156-57-0 Product: Tirapazamine
Synonym: GSK525762A; GSK-525762A; I-BET762; I-BET 762
Chemical Formula: C22H22ClN5O2
Appearance: Solid powderMedchemexpress
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).5-Lipoxygenase inhibitors
Solubility: Soluble in DMSO
Background Description: GSK 525762A is a small molecule inhibitor of the BET (Bromodomain and Extra-Terminal) family of bromodomain-containing proteins with potential antineoplastic activity.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/22588880
