Product Name: CPI-203
Chemical Name: (6S)-4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide
SMILES Code: ClC1=CC=C(C=C1)C2=N[C@@H](CC(N)=O)C3=NN=C(C)N3C4=C2C(C)=C(C)S4
CAS NO: 191114-48-4 Product: Guanfacine
Synonym: CPI203; CPI 203
Chemical Formula: C19H18ClN5OS
Appearance: Solid powderWeb Site click
Purity: 98% (this data is for the first batch)
Shipping Condition: Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition: Dry, dark and at 0 8211; 4 C for short term (days to weeks) or -20 C for long term (months to years).TRP Channel inhibitors
Solubility: Soluble in DMSO, not in water
Background Description: CPI203 is a novel potent, selective and cell permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 with an IC50 of ~37 nM. CPI203 enhances the antiproliferative effects of rapamycin on human neuroendocrine tumors.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/18708635
