Product Name: BX795 | PDK1/TBK1 inhibitor
Product Description: BX-795 is an aminopyrimidine-based, ATP-competitive inhibitor of PDK1, TBK1, and IKKe, with IC50 values of 11 nM, 6 nM, and 41 nM, respectively. [1, 2] BX-795 also potently inhibits ERK8, MNK2, Aurora B, Aurora C, and MARK3. [3] BX-795 inhibits both Thr30Medchemexpress
Chemical Formula: C23H26IN7O2S
Molecular Weight: 591.47
‘&“CAS NO: 1629268-00-3 ARS-853
Purity: 98%
Appearance: White
Chemical Name: N-(3-(5-iodo-4-(3-(thiophene-2-carboxamido)propylamino)pyrimidin-2-ylamino)phenyl)pyrrolidine-1-carboxamideReverse Transcriptase inhibitors
Solubility: Up to 100 mM in DMSO
Shipping Condition: The product is shipped in a glass vial at ambient temperature.
Storage Condition: For longer shelf life, store solid powder at 4oC desiccated, or store DMSO solution at -20oC.PubMed ID:http://www.ncbi.nlm.nih.gov/pubmed/23434473
